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CGS 15943
CAS No. 104615-18-1
CGS 15943 ( —— )
Catalog No. M23255 CAS No. 104615-18-1
CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.
Purity : >98% (HPLC)
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
| Size | Price / USD | Stock | Quantity |
| 5MG | 82 | In Stock |
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| 10MG | 120 | In Stock |
|
| 25MG | 201 | In Stock |
|
| 50MG | 300 | In Stock |
|
| 100MG | 448 | In Stock |
|
| 200MG | Get Quote | In Stock |
|
| 500MG | Get Quote | In Stock |
|
| 1G | Get Quote | In Stock |
|
Biological Information
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Product NameCGS 15943
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NoteResearch use only, not for human use.
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Brief DescriptionCGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.
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DescriptionCGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.
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Synonyms——
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PathwayEndocrinology/Hormones
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TargetAChR
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RecptorAdenosine A1?receptor;adenosine A2A receptor;adenosine A2B receptor;adenosine A3 receptor;p110γ;p110δ
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Research Area——
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Indication——
Chemical Information
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CAS Number104615-18-1
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Formula Weight285.7
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Molecular FormulaC13H8ClN5O
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Purity>98% (HPLC)
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SolubilityDMSO:12.22 mg/mL (42.77 mM; Need ultrasonic)
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SMILESC1=COC(=C1)C2=NN3C(=N2)C4=C(C=CC(=C4)Cl)N=C3N
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Chemical Name——
Shipping & Storage Information
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Storage(-20℃)
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ShippingWith Ice Pack
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Stability≥ 2 years
Reference
1.Gao Y, et al. CGS 15943, an adenosine A2 receptor antagonist, reduces cerebral ischemic injury in the Mongolian gerbil. Life Sci. 1994;55(3):PL61-5.
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