CGS 15943

CAS No. 104615-18-1

CGS 15943 ( —— )

Catalog No. M23255 CAS No. 104615-18-1

CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 82 In Stock
10MG 120 In Stock
25MG 201 In Stock
50MG 300 In Stock
100MG 448 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CGS 15943
  • Note
    Research use only, not for human use.
  • Brief Description
    CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.
  • Description
    CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    AChR
  • Recptor
    Adenosine A1?receptor;adenosine A2A receptor;adenosine A2B receptor;adenosine A3 receptor;p110γ;p110δ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    104615-18-1
  • Formula Weight
    285.7
  • Molecular Formula
    C13H8ClN5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:12.22 mg/mL (42.77 mM; Need ultrasonic)
  • SMILES
    C1=COC(=C1)C2=NN3C(=N2)C4=C(C=CC(=C4)Cl)N=C3N
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Gao Y, et al. CGS 15943, an adenosine A2 receptor antagonist, reduces cerebral ischemic injury in the Mongolian gerbil. Life Sci. 1994;55(3):PL61-5.
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