CGS 15943

CAS No. 104615-18-1

CGS 15943 ( —— )

Catalog No. M23255 CAS No. 104615-18-1

CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
5MG 82 In Stock
10MG 120 In Stock
25MG 201 In Stock
50MG 300 In Stock
100MG 448 In Stock
200MG Get Quote In Stock
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Biological Information

  • Product Name
    CGS 15943
  • Note
    Research use only, not for human use.
  • Brief Description
    CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.
  • Description
    CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor. In transfected CHO cells, its Ki for human A1, A2A, A2B, and A3 Adenosine Receptors are 3.5, 4.2, 16, and 50 nM , respectively.
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    AChR
  • Recptor
    Adenosine A1?receptor;adenosine A2A receptor;adenosine A2B receptor;adenosine A3 receptor;p110γ;p110δ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    104615-18-1
  • Formula Weight
    285.7
  • Molecular Formula
    C13H8ClN5O
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO:12.22 mg/mL (42.77 mM; Need ultrasonic)
  • SMILES
    C1=COC(=C1)C2=NN3C(=N2)C4=C(C=CC(=C4)Cl)N=C3N
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Gao Y, et al. CGS 15943, an adenosine A2 receptor antagonist, reduces cerebral ischemic injury in the Mongolian gerbil. Life Sci. 1994;55(3):PL61-5.
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